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Category: 7TM ReceptorsarrowPeptides (Cardiovascular)arrowUrotensin II Receptors
Cat.No. Product Name
2529 UFP 803
Price and Availability

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UFP 803

Biological Activity:

Urotensin II (UT) receptor ligand; behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays. Competitively antagonises UT-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by UT-II in mice in vivo.

Technical Data:

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M.Wt: 1061.24
Formula: C50H64N10O12S2
Storage: Desiccate at -20°C
CAS No: [879497-82-2]

Resources:

  • Certificate of Analysis / MSDS:

    Certificate of Analysis: View current batch
    Product/Material Safety Data Sheet: View current batch

    References:

    Camarda et al (2006) In vitro and in vivo pharmacological characterization of the novel UT receptor ligand [Pen5,DTrp7,Dab8]urotensin II(4-11) (UFP-803). Br.J.Pharmacol. 147 92.
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    Keywords: UFP 803, Peptides (Cardiovascular), Urotensin II (UT) Antagonist, UFP803, Tocris Bioscience

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