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Category: EnzymesarrowOxygenases/OxidasesarrowLipoxygenase
Cat.No. Product Name
0645 2-(1-Thienyl)ethyl 3,4-dihydroxybenzylidenecyanoacetate  
Price and Availability

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2-(1-Thienyl)ethyl 3,4-dihydroxybenzylidenecyanoacetate

Biological Activity:

Potent  inhibitor of 5-, 12-, and 15-lipoxygenase (IC50 values are 0.09, 0.013 and 0.5 μM respectively).

Technical Data:

Click here for more information on batch specific data
M.Wt: 315.34
Formula: C16H13NO4S
Storage: Desiccate at +4°C
Solubility: Soluble to 100 mM in DMSO and to 25 mM in Ethanol

Resources:

  • Certificate of Analysis / MSDS:

    Certificate of Analysis: View current batch
    Product/Material Safety Data Sheet: View current batch

    References:

    Cho et al (1991) Novel caffeic acid derivatives - extremely potent inhibitors of 12-lipoxygenase. J.Med.Chem. 34 1503.
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    Keywords: 2-(1-Thienyl)ethyl 3,4-dihydroxybenzylidenecyanoacetate, Oxygenases / Oxidases, 5-, 12-, 15-Lipoxygenase Inhibitor, 2(1-Thienyl)ethyl 3,4-dihydroxybenzylidenecyanoacetate, Tocris Bioscience

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