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Category: Cellular Processes and ComponentsarrowSignal TransductionarrowG Protein (Heterotrimeric)
Cat.No. Product Name
1884 [D-Trp7,9,10]-Substance P
Alternative name(s): GPAnt-2 analog
Price and Availability

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[D-Trp 7,9,10]-Substance P

Biological Activity:

Substance P analogue that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.

Technical Data:

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M.Wt: 1588.89
Formula: C79H105N21O13S
Storage: Desiccate at -20°C
CAS No: [89430-38-6]

Resources:

  • Certificate of Analysis / MSDS:

    Certificate of Analysis is currently unavailable on-line. Please contact Customer Service
    Product/Material Safety Data Sheet: View current batch

    References:

    Mukai et al (1992) G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J.Biol.Chem. 267 16237.
    View related products by Pharmacological Action or by Research Area

    Keywords: [D-Trp 7,9,10]-Substance P, Signal Transduction, Inhibits M1 ACh Receptor Activation Of Gq / 11, GPAnt-2 Analog, [DTrp 7,9,10]-Substance P, Tocris Bioscience

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