Rilmenidine Hemifuramate | Adrenergic Receptors | A2 Agonist. Also I1 Ligand

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Cat.No.	Product Name
0790	Rilmenidine hemifuramate

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Rilmenidine hemifuramate

Chemical Name: 2-[N-(Dicyclopropylmethyl)amino]oxazoline hemifuramate

Biological Activity:

I₁-imidazoline binding site selective ligand and α₂-adrenoceptor agonist. Possesses greater I₁ vs α₂selectivity than the prototypical compound, clonidine.

Technical Data:

M.Wt:	238.29
Formula:	C₁₀H₁₆N₂O.½C₄H₄O₄
Storage:	Store at RT
Solubility:	Soluble to 25 mM in DMSO and to 25 mM in Ethanol
CAS No:	[54187-04-1]

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References:

Bricca et al (1989) Rilmenidine selectivity for imidazoline receptors in human brain. Eur.J.Pharmacol. 163 373. Michel and Ernsberger (1992) Keeping an eye on the I site: imidazoline-preferring receptors. TiPS 13 369. Bricca et al (1994) Human brain imidazoline receptors: Further characterisation with [³H] clonidine. Eur.J.Pharmacol.Mol.Pharmacol.Sect. 266 25. Mammoto et al (1996) Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs. Br.J.Pharmacol. 117 1744.

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Keywords: Rilmenidine Hemifuramate, Adrenergic Receptors, A2 Agonist. Also I1 Ligand , Tocris Bioscience

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Adrenoceptor Pharmacology
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