2-[1-(4-Piperonyl)piperazinyl]benzothiazole | 5-HT Receptors | 5-HT4 Agonist. Also 5-HT3 Antagonist | 2[1-(4-Piperonyl)piperazinyl]benzothiazole

Category:

Cat.No.	Product Name
0736	2-[1-(4-Piperonyl)piperazinyl]benzothiazole

Price and Availability

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2-[1-(4-Piperonyl)piperazinyl]benzothiazole

Biological Activity:

5-HT₄ receptor agonist with moderate activity as a 5-HT₃ antagonist. Has no affinity at 5-HT₁ or dopamine D₂ receptors. Potential gastrokinetic agent.

Technical Data:

M.Wt:	353.44
Formula:	C₁₉H₁₉N₃O₂S
Storage:	Store at RT
Solubility:	Soluble to 10 mM in DMSO

Resources:

Certificate of Analysis / MSDS:

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Product/Material Safety Data Sheet: View current batch

References:

Monge et al (1994) Synthesis of 2-piperazinybenzothiazole and 2-piperazinylbenzoxazole derivatives with 5-HT₃ antagonist and 5-HT₄ agonist properties. J.Med.Chem. 37 1320.

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Keywords: 2-[1-(4-Piperonyl)piperazinyl]benzothiazole, 5-HT Receptors, 5-HT4 Agonist. Also 5-HT3 Antagonist, 2[1-(4-Piperonyl)piperazinyl]benzothiazole, Tocris Bioscience

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