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Category:
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7TM Receptors Cannabinoid ReceptorsNon-selective CB1/CB2
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Cat.No.
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Product Name
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2680 |
O-2545 hydrochloride
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Price and Availability
Click here for full price details of
O-2545
Other Information:
Sold
under licence
from VCU-IPF
DEA controlled substance.
Please consult your local
office for further information.
Canadian customers require a CDSA import
permit
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Chemical Name:
(6aR,10aR)-6a,7,10,10a-Tetrahydro-3-[5-(1H-imidazol-1-y
l)-1,1-dimethylpentyl]-6,6,9-trimethyl-6H-dibenzo[b,d]p
yran-1-ol hydrochloride |
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Biological Activity:
High affinity, water-soluble CB1/CB2
receptor agonist (Ki values are 1.5 and 0.32 nM for CB1
and CB2 receptors respectively). Active in vivo following i.v. and
i.c.v. administration.
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Martin et al
(2006) Pharmacological characterization of novel water-soluble cannabinoids.
J.Pharmacol.Exp.Ther. 318 1230.
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View related products by Pharmacological Action
or by Research Area
Keywords: O-2545, Cannabinoid Receptors, High Affinity, Water-soluble CB1 / CB2 Agonist, O2545, Tocris Bioscience
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