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Category: 7TM ReceptorsarrowOpioid ReceptorsarrowMiscellaneous Opioids
Cat.No. Product Name
0677 Naltrexone hydrochloride  
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Naltrexone hydrochloride

Other Information:

Controlled in Australia under the Standard for the Uniform Scheduling of Drugs and Poisons; Schedule 4 drug .

Please consult your local office for further information
Chemical Name: (5a)-17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydromorph inan-6-one hydrochloride

Biological Activity:

Opioid antagonist.

Technical Data:

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M.Wt: 377.87
Formula: C20H23NO4.HCl
Storage: Store at RT
Solubility: Soluble to 100 mM in Water
CAS No: [16676-29-2]

Resources:

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    References:

    Zukin et al (1982) Naltrexone-induced opiate receptor supersensitivity. Brain Res. 245 285. Tempel et al (1982) Supersensitivity of brain opiate receptor subtypes after chronic naltrexone treatment. Life Sci. 31 1401. Gold et al (1982) Naltrexone, opiate addiction, and endorphins. Med.Res.Rev. 2 211.

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    Keywords: Naltrexone Hydrochloride, Opioid Receptors, Broad Spectrum Opioid Antagonist, Tocris Bioscience

    Literature in this Area
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    Opioid Receptors
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