Naloxonazine Dihydrochloride | Opioid Receptors | Selective µ1 Antagonist

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Cat.No.	Product Name
0591	Naloxonazine dihydrochloride

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Naloxonazine dihydrochloride

Chemical Name: Bis-[5-a-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)-morph inan-6-ylidene] hydrazine dihydrochloride

Biological Activity:

Potent opioid antagonist, selective for m₁ receptors.

Technical Data:

M.Wt:	723.69
Formula:	C₃₈H₄₂N₄O₆.2HCl
Storage:	Store at RT
Solubility:	Soluble to 25 mM in Water
Purity:	>98%
CAS No:	[82824-01-9]

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References:

Paul et al (1988) Differential blockade by naloxonazine of two μ opiate actions: analgesic and inhibition of gastrointestinal transit. Eur.J.Pharmacol. 149 403.

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Keywords: Naloxonazine Dihydrochloride, Opioid Receptors, Selective µ1 Antagonist, Tocris Bioscience

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Scientific Reviews

Opioid Receptors
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