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Category:
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7TM Receptors P2Y Receptors Antagonists
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Cat.No.
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Product Name
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2402 |
MRS 2211
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Price and Availability
Click here for full price details of
MRS 2211
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Chemical Name:
2-[(2-Chloro-5-nitrophenyl)azo]-5-hydroxy-6-methyl-3-[(
phosphonooxy)methyl]-4-pyridinecarboxaldehyde disodium
salt |
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Biological Activity:
Competitive
P2Y13 receptor antagonist (pIC50 = 5.97) that displays
> 20-fold selectivity over P2Y1 and P2Y12 receptors.
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Kim et al (2005) Synthesis of
pyridoxal phosphate derivatives with antagonist activity at the P2Y13
receptor. Biochem.Pharmacol. 70 266. Kugelgen (2006)
Pharmacological profiles of cloned mammalian P2Y-receptor subtypes.
Pharmacol.Ther. 110 415.
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Keywords: MRS 2211, P2Y Receptors, Competitive P2Y13 Antagonist, MRS2211, Tocris Bioscience
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