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Category: 7TM Receptorsarrow5-HT Receptorsarrow5-HT2 Receptorsarrow5-HT2C
Cat.No. Product Name
0941 MK 212 hydrochloride  
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MK 212 hydrochloride
Chemical Name: 6-Chloro-2-(1-piperazinyl)pyrazine hydrochloride

Biological Activity:

5-HT2C serotonin receptor agonist.

Technical Data:

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M.Wt: 235.12
Formula: C8H11CIN4.HCl
Storage: Store at RT
Solubility: Soluble to 50 mM in Water
Purity: >99%
CAS No: [64022-27-1]

Resources:

  • Certificate of Analysis / MSDS:

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    References:

    Conn and Sanders-Bush (1987) Relative efficacies of piperazines at the phosphoinositide hydrolysis-linked serotonergic (5-HT2 and 5-HT1C) receptors. J.Pharmacol.Exp.Ther. 242 552. Lee et al (1992) Effect of the serotonin agonist, MK-212, on body temperature in schizophrenia. Biol.Psychiatry 31 460. Hemrick-Luecke and Fuller (1996) Involvement of 5-HT2A receptors in the elevation of rat serum corticosterone concentration by quipazine and MK-212. Eur.J.Pharmacol. 311 207.

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    Keywords: MK 212 Hydrochloride, 5-HT Receptors, 5-HT2C Agonist, MK212 Hydrochloride, Tocris Bioscience

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