M871 | Peptides (Gastrointestinal) | Selective GalR2 Antagonist | Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide

Category:

7TM Receptors

Peptides (Gastrointestinal)

Galanin Receptors

Cat.No.

Product Name

2698

M871

Alternative name(s):

Galanin-(2-13)-Glu-His-(Pro)₃-(Ala-Leu)₂-Ala-amide

Price and Availability

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M871

Biological Activity:

Selective galanin GalR2 receptor antagonist (K_i values are 13.1 and 420 nM for GalR2 and GalR1 receptors respectively). Blocks the pro-nociceptive effect of GalR2 receptor agonists.

Technical Data:

M.Wt:	2287.64
Formula:	C₁₀₈H₁₆₃N₂₇O₂₈
Storage:	Desiccate at -20°C
CAS No:	[908844-75-7]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Sollenburg et al (2006) M871 - a novel peptide antagonist selectively recognizing the galanin receptor type 2. Int.J.Pept.Res.Ther. 12 115. Jimenez-Andrade et al (2006) Activation of peripheral galanin receptors: differential effects on nociception. Pharmacol.Biochem.Behav. 85 273.

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Keywords: M871, Peptides (Gastrointestinal), Selective GalR2 Antagonist, Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide, Tocris Bioscience

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