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Category:
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7TM Receptors Peptides (Gastrointestinal)Galanin Receptors
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Cat.No.
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Product Name
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2697 |
M617
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| Alternative name(s): |
Galanin(1-13)-Gln14-bradykinin(2-9)amide |
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Price and Availability
Click here for full price details of
M617
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Biological Activity:
Selective galanin GalR1 receptor agonist (Ki
values are 0.23 and 5.71 nM for GalR1 and GalR2 receptors respectively).
Enhances food consumption in rats following i.c.v. administration and reduces
CAP-induced inflammatory pain.
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Lundstrom et al
(2005) A galanin receptor subtype 1 specific agonist. Int.J.Pept.Res.Ther. 11
17. Mazarati et al (2006) Regulation of kindling epileptogenesis
by hippocampal galanin type 1 and type 2 receptors: the effects of
subtype-selective agonists and the role of G-protein-mediated signaling.
J.Pharmacol.Exp.Ther. 318 700. Jimenez-Andrade et al
(2006) Activation of peripheral galanin receptors: differential effects on
nociception. Pharmacol.Biochem.Behav. 85 273.
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Keywords: M617, Peptides (Gastrointestinal), Selective GalR1 Agonist, Galanin(1-13)-Gln14-bradykinin(2-9)amide, Tocris Bioscience
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