Iodophenpropit Dihydrobromide | Histamine Receptors | Potent, Selective H3 Antagonist

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Cat.No.	Product Name
0779	Iodophenpropit dihydrobromide

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Iodophenpropit dihydrobromide

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Sold with the permission of SCI, Amsterdam

Chemical Name: N-[2-(4-Iodophenyl)ethyl]-S-[3-(4(5)-imidazolyl)propyl] isothiourea dihydrobromide

Biological Activity:

Selective H₃ antagonist with high affinity.

Technical Data:

M.Wt:	576.13
Formula:	C₁₅H₁₉IN₄S.2HBr
Storage:	Desiccate at +4°C
Solubility:	Soluble to 25 mM in Water
CAS No:	[143407-29-8]

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References:

Jansen et al (1992) The first radiolabelled histamine H₃ receptor antagonist, [¹²⁵I]iodophenpropit: saturable and reversible binding to rat cortex membranes. Eur.J.Pharmacol. 217 203. Menge et al (1992) Synthesis of S-[3-(4(5)-imidazolyl)propyl]-N-[2-(4-[¹²⁵I]-iodophenylethyl]isothiourea sulfate [¹²⁵I]-iodophenpropit), a new probe for histamine H₃ receptor binding sites. J.Labelled Comp.Radiopharm. XXXI 10 781. Jansen et al (1994) Characterisation of the binding of the first selective radiolabelled histamine H₃ receptor antagonist, [¹²⁵I]-iodophenpropit, to rat brain. Br.J.Pharmacol. 113 355.

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Keywords: Iodophenpropit Dihydrobromide, Histamine Receptors, Potent, Selective H3 Antagonist, Tocris Bioscience

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