GR 82334 | Peptides (Neuropeptides) | Tachykinin NK1 Receptor Antagonist | GR82334

Category:

Cat.No.	Product Name
1670	GR 82334

Price and Availability

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GR 82334

Other Information:

Sold for research purposes under agreement from GlaxoSmithKline

Biological Activity:

Tachykinin NK₁ receptor antagonist.

Technical Data:

M.Wt:	1386.57
Formula:	C₆₉H₉₁N₁₅O₁₆
Storage:	Desiccate at -20°C
CAS No:	[129623-01-4]

Resources:

Certificate of Analysis / MSDS:

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References:

Hagan et al (1991) A spirolactam conformationally-constrained analogue of physalaemin which is a peptidase-resistant, selective neurokinin NK-1 receptor antagonist. Br.J.Pharmacol. 102 168P. Lecci et al (1992) Effect of the NK-1 receptor antagonist GR 82,334 on reflexly-induced bladder contractions. Life Sci. 51 277. Guo et al (1995) Pharmacological characterisation of GR82334, a tachykinin NK₁ receptor antagonist, in the isolated spinal cord of the neonatal rat. Eur.J.Pharmacol. 281 49.

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Keywords: GR 82334, Peptides (Neuropeptides), Tachykinin NK1 Receptor Antagonist, GR82334, Tocris Bioscience

Literature in this Area

Scientific Reviews

Tachykinin Receptor Compounds
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