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Category: 7TM ReceptorsarrowPeptides (Neuropeptides)arrowTachykinin ReceptorsarrowNK-1 Receptor
Cat.No. Product Name
1669 GR 73632
Price and Availability

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GR 73632

Other Information:

Sold for research purposes under agreement from GlaxoSmithKline

Biological Activity:

Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea-pig vas deferens). Active in vivo.

Technical Data:

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M.Wt: 766.01
Formula: C40H59N7O6S
Storage: Desiccate at -20°C
CAS No: [133156-06-6]

Resources:

  • Certificate of Analysis / MSDS:

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    References:

    Hall and Morton (1991) Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation. Ann.N.Y.Acad.Sci. 632 404. Meini et al (1995) GR 73,632 and [glu(OBzl)11]substance P are selective agonists for the septide-sensitive tachykinin NK1 receptor in the rat urinary bladder. Neuropeptides 28 99. Sakurada et al (1999) Spinal actions of GR73632, a novel tachykinin NK1 receptor agonist. Peptides 20 301.
    View related products by Pharmacological Action or by Research Area

    Keywords: GR 73632, Peptides (Neuropeptides), Potent, Selective NK1 Agonist, GR73632, Tocris Bioscience

    Literature in this Area
    Scientific Reviews
    Tachykinin Receptor Compounds
    Download PDF
    Tocris is to be congratulated for continuing to meet the current demand for a rapid and reliable source of high-quality compounds that are urgently needed as pharmacological tools by a growing international population of cannabinoid researchers..”
    Researcher, University of Aberdeen, UK
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