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Category: 7TM Receptorsarrow5-HT Receptorsarrow5-HT1 Receptorsarrow5-HT1B
Cat.No. Product Name
0458 5-Carboxamidotryptamine maleate  
Alternative name(s): AH-21467
5-CT
Price and Availability

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5-Carboxamidotryptamine maleate

Biological Activity:

5-HT1 agonist with high affinity at 5-HT1A, 5-HT1B , 5-HT1D, 5-ht5 and 5-HT7 receptors.

Technical Data:

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M.Wt: 319.32
Formula: C11H13N3O.C4H4O4
Storage: Desiccate at +4°C
Solubility: Soluble to 100 mM in Water
Purity: >99%
CAS No: [74885-09-9]

Resources:

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    References:

    Beer et al (1992) An investigation of the 5-HT1D receptor binding affinity of 5-hydroxytryptamine, 5-carboxyamidotryptamine and sumatriptan in the central nervous system of seven species. Eur.J.Pharmacol. 213 193. Zifa and Fillion (1992) 5-Hydroxytryptamine receptors. Pharmacol.Rev. 44 402. Nowak et al (1993) [3H]-5-carboxamidotryptamine labels 5HT1D binding sites in bovine substantia nigra. Br.J.Pharmacol. 109 1206. Wood et al (2000) Antagonist activity of meta-chlorophenylpiperazine and partial agonist activity of 8-OH-DPAT at the 5-HT7 receptor. Eur.J.Pharmacol. 396 1.

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    Keywords: 5-Carboxamidotryptamine Maleate, 5-HT Receptors, 5-HT1 Agonist. Also Has High Affinity For 5-ht5A & 5-HT7, AH-21467, 5-CT, 5Carboxamidotryptamine Maleate, Tocris Bioscience

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