Category:
Nuclear Receptors Retinoic Acid Receptors
Cat.No.
Product Name
2554
CD 1530
Price and Availability
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CD 1530
Chemical Name:
4-(6-Hydroxy-7-tricyclo[3.3.1.13,7]dec-1-yl-2-naphthale
nyl)benzoic acid
Biological Activity:
Potent and selective RAR γ receptor
agonist (Ki values are 150, 1500 and 2750 nM for RAR γ , RAR β and RAR α receptors
respectively). Activates transcriptional activity (AC50 = 1.8 nM).
Technical Data:
Resources:
Certificate of Analysis / MSDS:
For specific/earlier batch please select: 1
For specific/earlier batch please select: 1
References:
Thacher et al
(2000) Therapeutic applications for ligands of retinoid receptors.
Curr.Pharmaceut.Des. 6 25.
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Keywords: CD 1530, Retinoic Acid Receptors, Potent & Selective RARg Agonist, CD1530, Tocris Bioscience
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