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Category: 7TM ReceptorsarrowDopamine ReceptorsarrowD2-like ReceptorsarrowAgonists
Cat.No. Product Name
0427 Bromocriptine mesylate  
Price and Availability

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Bromocriptine mesylate
Chemical Name: (5'a)-2-Bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-meth ylpropyl)ergotaman-3',6',18-trione mesylate

Biological Activity:

Selective D2-like dopamine receptor agonist (Ki values are ~ 8, ~ 5, ~ 290, ~ 440 and ~ 450 nM for D2, D3, D4, D1 and D5 receptors respectively).

Technical Data:

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M.Wt: 750.7
Formula: C32H40BrN5O5.CH3SO3H
Storage: Store at RT
Solubility: Soluble to 5 mM in Ethanol and to 10 mM in DMSO
CAS No: [22260-51-1]

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    References:

    Traub et al (1985) The effects of chronic bromocriptine treatment on behaviour and dopamine receptor binding in the rat striatum. Eur.J.Pharmacol. 118 147. Lieberman and Goldstein (1985) Bromocriptine in Parkinson disease. Pharmacol.Rev. 37 217. Aubner et al (1990) Bromocriptine produces decreases in cocaine self-administration in the rat. Neuropsychopharmacology 3 101. Seeman and Van Tol (1994) Dopamine receptor pharmacology. TiPS 15 264.
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    Keywords: Bromocriptine Mesylate, Dopamine Receptors, Selective D2-like Agonist, Tocris Bioscience
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