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Category:
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7TM Receptors Peptides (Neuropeptides)NPY Receptors
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Cat.No.
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Product Name
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2177 |
BVD 10
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Price and Availability
Click here for full price details of
BVD 10
Other Information:
Sold under licence
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Biological Activity:
Highly
selective NPY Y1 receptor antagonist. Ki values are 25.7,
1420, 2403 and 7100 nM at Y1, Y2, Y4 and Y5
receptors respectively. Devoid of agonist activity at Y4 receptors.
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
Certificate of Analysis is currently unavailable on-line. Please contact Customer Service
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References:
Balasubramaniam et al (2001) Highly selective and potent neuropeptide
Y (NPY) Y1 receptor antagonists based on [Pro30, Tyr32,
Leu34]NPY(28-36)-NH2 (BW1911U90). J.Med.Chem. 44
1479. Jois and Balasubramaniam (2003) Conformation of neuropeptide Y
receptor antagonists: structural implications in receptor selectivity. Peptides
24 1035.
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View related products by Pharmacological Action
or by Research Area
Keywords: BVD 10, Peptides (Neuropeptides), Highly Selective Y1 Antagonist; Devoid Of Y4 Agonist Activity, BVD10, Tocris Bioscience
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