|
Category:
|
7TM Receptors Peptides (Gastrointestinal)Apelin Receptors
|
|
Cat.No.
|
Product Name
|
|
2420 |
[Pyr1]-Apelin-13
|
| Alternative name(s): |
[pGlu1]-Apelin-13 |
|
|
Price and Availability
Click here for full price details of
[Pyr1]-Apelin-13
|
|
|
|
|
Biological Activity:
Highly
potent proglutamyl form of apelin-13. Endogenous ligand for apelin APJ receptor
(EC50 = 0.37 nM) that displays potent vascular effects in vivo.
|
Technical Data:
|
|
|
Resources:
|
|
Certificate of Analysis / MSDS:
|
References:
Tatemoto et al (1998) Isolation
and characterization of a novel endogenous peptide ligand for the human APJ
receptor. Biochem.Biophys.Res.Comm. 251 471. Katugampola et al (2001) [125I]-(Pyr1)Apelin-13
is a novel radioligand for localizing the APJ orphan receptor in human and rat
tissues with evidence for a vasoconstrictor role in man. Br.J.Pharmacol. 132
1255. Kagiyama et al (2005) Central and peripheral cardiovascular
actions of apelin in conscious rats. Regul.Pept. 125 55.
|
|
View related products by Pharmacological Action
or by Research Area
Keywords: [Pyr1]-Apelin-13, Peptides (Gastrointestinal), Potent Peptide Agonist For APJ Receptor, [pGlu1]-Apelin-13, Tocris Bioscience
|
|
Dedicated Customer Service
At Tocris we understand that customer service means more than just taking orders, we are here to act in partnership with you and to help you further your research. We do our best to ensure that your purchasing experience at Tocris is quick and effortless.
We are committed to making sure that over 99% of our products are in stock and in every case Tocris provides same day shipping of orders. Our friendly and efficient team delivers top quality support time after time.
|
|
