R&D Systems Inc. Tocris Bioscience Boston Biochem

Androgen Receptors

More Information »Androgen receptors (ARs) (dihydrotestosterone receptors) are nuclear hormone receptors of the NR3C class, which includes mineralocorticoid, progesterone and glucocorticoid receptors. ARs are expressed in bone marrow, mammary gland and prostate tissues.

Androgen Receptor Products

Agonists
Cat.No.
Product Name / Activity
3812 Cl-4AS-1
Steroidal androgen receptor agonist
2822 Testosterone
Endogenous androgen receptor agonist
Antagonists
Cat.No.
Product Name / Activity
3389 Bicalutamide
Non-steroidal androgen receptor antagonist
4094 Flutamide
Non-steroidal androgen receptor antagonist
1759 Nilutamide
Androgen receptor antagonist. Orally active
3923 PF 998425
Non-steroidal androgen receptor antagonist
Modulators
Cat.No.
Product Name / Activity
3813 TFM-4AS-1
Selective androgen receptor modulator (SARM)
Other
Cat.No.
Product Name / Activity
4946 AIM 100
Potent and selective Ack1 inhibitor
4626 Andrographolide
Inhibits NFκB; blocks androgen receptor (AR) expression
3293 Finasteride
Type II 5α-reductase inhibitor
3572 GSK 650394
Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
4396 Piperlongumine
Induces apoptosis; depletes androgen receptors in prostate cancer cells
2968 Spironolactone
Antiandrogen; inhibits steroid hormone biosynthesis. Also MR antagonist
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