R&D Systems Inc. Tocris Bioscience Boston Biochem

Purinergic (P2X) Receptors

More Information »P2X receptors are members of the ligand-gated ion channel family that open in response to extracellular ATP. Each receptor is made up of a trimer of subunits (P2X1-7) all of which share the common structure of two transmembrane domains.

Purinergic (P2X) Receptors Products

Agonists
Cat.No.
Product Name / Activity
3245 ATP disodium salt
P2 purinergic agonist
4080 ATPγS tetralithium salt
P2 agonist; ATP (Cat. No. 3245) analog
3312 BzATP triethylammonium salt
P2X7 agonist. Also P2X1 and P2Y1 partial agonist
3209 α,β-Methyleneadenosine 5'-triphosphate trisodium salt
P2-purinoceptor agonist
1062 2-Methylthioadenosine triphosphate tetrasodium salt
P2 purinergic agonist
Antagonists
Cat.No.
Product Name / Activity
2972 A 438079 hydrochloride
Competitive P2X7 antagonist
3701 A 740003
Potent and selective P2X7 antagonist
4473 A 804598
Potent and selective P2X7 antagonist
4232 A 839977
Potent P2X7 antagonist
3323 AZ 10606120 dihydrochloride
Potent P2X7 receptor antagonist
3317 AZ 11645373
Potent and selective human P2X7 antagonist
3579 5-BDBD
Potent P2X4 receptor antagonist
0845 Evans Blue tetrasodium salt
Selective P2X purinergic antagonist
1277 KN-62
Non-competitive P2X7 antagonist
1240 NF 023
Selective, competitive P2X1 antagonist
2548 NF 110
Potent P2X3 antagonist
2450 NF 157
Selective P2Y11/P2X1 antagonist
1199 NF 279
Potent and selective P2X1 antagonist
1391 NF 449
Highly selective P2X1 antagonist
0625 PPADS tetrasodium salt
P2 purinergic antagonist
0683 iso-PPADS tetrasodium salt
P2X antagonist
1309 PPNDS
Potent, selective P2X1 antagonist
2188 Ro 0437626
Selective P2X1 antagonist
4391 Ro 51
Potent P2X3, P2X2/3 antagonist
3052 RO-3
Selective P2X3 and P2X2/3 antagonist
2931 Spinorphin
Potent P2X3 antagonist
1472 Suramin hexasodium salt
Non-selective P2 antagonist
4386 TC-P 262
Selective P2X3, P2X2/3 antagonist
2464 TNP-ATP triethylammonium salt
Potent, selective P2X antagonist
Modulators
Cat.No.
Product Name / Activity
3385 GW 791343 hydrochloride
P2X7 allosteric modulator
1260 Ivermectin
Positive allosteric modulator for P2X4 receptor
4922 Purotoxin 1
Potent P2X3 modulator
Other
Cat.No.
Product Name / Activity
5157 DMNPE-caged ATP diammonium salt
Caged ATP
5156 Ivermectin B1a-d2
Deuterated ivermectin B1a (Cat. No. 1260)
1203 MRS 2219
Potentiates P2X1-mediated responses
Related Categories

Quick Order

Find multiple products by catalog number

divider line

Pain Research Product Guide

Pain Research Guide

Highlights over 280 products for Pain research. Request copy or view PDF today.

divider line

P2 Receptors Review

Purinergic Receptor Review

Written by Kenneth Jacobson, an expert in the field. Request a copy or view PDF today.

divider line

New Product Guide

NPG

Highlights over 130 new products added in the second half of 2013. Request a copy or view PDF today.

divider line

Tocris Events

Win $1,000 Product Credit

Experimental Biology

Experimental Biology

April 26 - 30, 2014

San Diego CA, USA

Booth Number: 918