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Voltage-gated Calcium Channels (CaV)
Blockers
Cat.No. |
Product Name / Activity |
| 2799 | ω-Agatoxin IVA |
| Ca2+ channel blocker (P-type) | |
| 2802 | ω-Agatoxin TK |
| Ca2+ channel blocker (P/Q-type) | |
| 2571 | Amlodipine besylate |
| Ca2+ channel blocker (L-type) | |
| 1545 | (R)-(+)-Bay K 8644 |
| Ca2+-channel blocker (L-type) | |
| 3934 | Benidipine hydrochloride |
| Calcium channel blocker | |
| 4117 | Bepridil hydrochloride |
| Non-selective calcium channel blocker | |
| 2629 | Cilnidipine |
| Ca2+ channel blocker (dual L/N-type) | |
| 1085 | ω-Conotoxin GVIA |
| Ca2+ channel blocker (N-type) | |
| 1084 | ω-Conotoxin MVIIC |
| Ca2+ channel blocker (N, P and Q-type) | |
| 0685 | Diltiazem hydrochloride |
| Ca2+ channel blocker (L-type) | |
| 3733 | Efonidipine hydrochloride monoethanolate |
| Ca2+ channel blocker (L- and T-type) | |
| 2960 | Felodipine |
| Ca2+ channel blocker (L-type) | |
| 0522 | Flunarizine dihydrochloride |
| Dual Na+/Ca2+ channel (T-type) blocker | |
| 2004 | Isradipine |
| Ca2+ channel blocker (L-type) | |
| 3086 | L-651,582 |
| Ca2+ channel blocker | |
| 2959 | Lercanidipine hydrochloride |
| Ca2+ channel blocker (L-type) | |
| 0840 | Loperamide hydrochloride |
| Ca2+ channel blocker (HVA) (L/N-type) | |
| 2198 | Mibefradil dihydrochloride |
| Ca2+ channel blocker (T-type) | |
| 4507 | ML 218 hydrochloride |
| Ca2+ channel blocker (T-type) | |
| 1075 | Nifedipine |
| Ca2+ channel blocker (L-type) | |
| 1124 | (R)-(-)-Niguldipine hydrochloride |
| Ca2+ channel blocker (L-type). Less active enantiomer of Cat. No. 1123 | |
| 1123 | (S)-(+)-Niguldipine hydrochloride |
| Ca2+ channel blocker (L-type) | |
| 0600 | Nimodipine |
| Ca2+ channel blocker (L-type) | |
| 0601 | Nitrendipine |
| Ca2+ channel blocker (L-type) | |
| 2268 | NNC 55-0396 dihydrochloride |
| Highly selective Ca2+ channel blocker (T-type) | |
| 3552 | PD 173212 |
| Potent N-type Ca2+ channel blocker | |
| 4665 | ProTx I |
| CaV3.1 channel blocker; also inhibits NaV1.8 and KV2.1 | |
| 1439 | Ruthenium Red |
| Non-selective Ca2+ channel blocker (N- and P-type) | |
| 2945 | SNX 482 |
| Potent and selective CaV2.3 blocker (R-type) | |
| 1806 | SR 33805 oxalate |
| Ca2+ channel blocker; binds allosterically to distinct site on L-type channels | |
| 0654 | Verapamil hydrochloride |
| Ca2+ channel blocker (L-type) | |
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