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Adrenergic β3 Receptors
More Information »The adrenergic β3 receptor (β3-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β1 and β2. They are located primarily in the small intestine, adipose tissue and vascular endothelium.
Adrenergic β3 Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 0948 | BRL 37344, sodium salt |
| β3 agonist | |
| 1134 | CGP 12177 hydrochloride |
| β3 partial agonist. β1/β2 antagonist. | |
| 1499 | CL 316243 disodium salt |
| Highly selective β3 agonist | |
| 0929 | ICI 215,001 hydrochloride |
| β3 agonist | |
| 2197 | L-755,507 |
| Very potent and selective β3 partial agonist | |
| 2242 | Octopamine hydrochloride |
| Invertebrate biogenic amine: activates β3 adrenoceptors | |
| 0994 | Pindolol |
| β3 partial agonist | |
| 1060 | (S)-(-)-Pindolol |
| β3 partial agonist. More active enantiomer of pindolol (Cat. No. 0994) | |
| 3986 | SR 58611A hydrochloride |
| β3 agonist; displays anxiolytic and antidepressant effects | |
| 2154 | ZD 2079 |
| β3-adrenoceptor agonist | |
| 0930 | ZD 7114 hydrochloride |
| β3 agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 2760 | L-748,337 |
| Selective β3 antagonist | |
| 1511 | SR 59230A hydrochloride |
| Potent and selective β3 antagonist | |
Ligand Sets |
|
Cat.No. |
Product Name / Activity |
| 1873 | β-Adrenoceptor Agonist Tocriset™ |
| Selection of 3 β-adrenoceptor agonists (Cat. Nos. 0948, 1747 and 1660) | |
| 1874 | β-Adrenoceptor Antagonist Tocriset™ |
| Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511) | |
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