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M2 Receptors
More Information »M2 receptors are members of the G-protein-coupled receptor (GPCR) family which are found mostly bound to Gi proteins, generally leading to inhibitory effects. They are one of five muscarinic receptors that act to control the metabotropic functions of acetylcholine in the CNS.
M2 Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 0382 | Arecaidine but-2-ynyl ester tosylate |
| Muscarinic agonist | |
| 0383 | Arecaidine propargyl ester tosylate |
| Muscarinic agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 1105 | AF-DX 116 |
| Selective M2 antagonist | |
| 1345 | AF-DX 384 |
| Potent M2/M4 antagonist | |
| 2292 | AQ-RA 741 |
| Selective, high affinity M2 antagonist | |
| 1425 | (S)-(+)-Dimethindene maleate |
| M2-selective antagonist | |
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