Cytochrome P450

More Information »Cytochrome P450 (CYP450) enzymes are a diverse group of catalysts that contains 57 members in humans. CYPs are usually membrane-bound and are localized to the inner mitochondrial or endoplasmic reticular membrane. CYPs have oxygenase activity.

Cytochrome P450 Products

Inhibitors
Cat.No.	Product Name / Activity
3388	Anastrozole
	Potent aromatase (CYP19) inhibitor
4096	Clotrimazole
	Cytochrome P450 inhibitor; antifungal
3759	Exemestane
	Steroidal aromatase (CYP19) inhibitor
1103	Ketoconazole
	Cytochrome P450c17 inhibitor
4382	Letrozole
	Potent, reversible non-steroidal aromatase inhibitor
2705	Liarozole hydrochloride
	Cytochrome P450 (CYP26) inhibitor; blocks retinoic acid metabolism
3292	Metyrapone
	Cytochrome P450 inhibitor
2583	Omeprazole
	CYP2C19, CYP2C9 and CYP3A inhibitor. Also H⁺,K⁺-ATPase inhibitor
4252	PF 4981517
	Selective CYP3A4 inhibitor
1509	TMS
	Cytochrome P450 1B1 inhibitor
3278	YM 511
	Potent aromatase (CYP19) inhibitor
Substrates
Cat.No.	Product Name / Activity
4815	3-Cyano-7-ethoxycoumarin
	Fluorescent cytochrome P450 substrate
3276	Mephenytoin
	CYP2C19 substrate. Anticonvulsant