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Estrogen (GPR30) Receptors
More Information »The GPR30 receptor is an orphan G-protein-coupled receptor that has recently been shown to bind estrogen and cause estrogen-mediated adenylyl cyclase stimulation. GPR30 is widely distributed in neural, breast cancer, placental, heart, ovarian, prostate and hepatic tissue.
Estrogen (GPR30) Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 2824 | β-Estradiol |
| Endogenous ER agonist | |
| 3577 | G-1 |
| Potent and selective GPR30 agonist | |
| 1110 | Genistein |
| GPR30 agonist. Also tyrosine kinase inhibitor | |
| 1047 | ICI 182,780 |
| High affinity GPR30 agonist | |
| 1125 | Quercetin |
| GPR30 agonist. Also non-selective PI 3-kinase inhibitor | |
| 0999 | Tamoxifen citrate |
| High affinity GPR30 agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 3678 | G-15 |
| High affinity and selective GPR30 antagonist | |
| 4759 |
G-36
|
| Selective GPR30 antagonist | |
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7-TM Receptor Signaling
Written by T. Kenakin et al
'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy
Estrogen Pathway
Estrogen controls many cellular processes including growth, differentiation and function of the reproductive system. View pathway or download PDF today.
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