Cat. No. 2710
Chemical Name: 2-[4-[[3-(4-Bromophenyl)-1-oxo-2-pr
Biological ActivityHeparanase inhibitor (IC50 = 0.4 μM) that displays no major inhibition of human cytochrome P450 isoenzymes (IC50 > 30 μM). Exhibits antiangiogenic properties in vitro (IC50 = 1 μM).
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Courtney et al (2005) Furanyl-1,3-thiazol-2-yl and benzoxazol-5-yl acetic acid derivates: novel classes of heparanase inhibitor. Bioorg.Med.Chem.Letts. 15 2295.
McKenzie (2007) Heparanase: a target for drug discovery in cancer and inflammation. Br.J.Pharmacol. 151 1. PMID: 17339837.
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Keywords: OGT 2115, supplier, Antiangiogenic, Heparanase, inhibitors, Antiangiogenics, Glycosylases, Carbohydrate, Metabolism, OGT2115
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May 2-6, 2014
Booth Number: 523