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PSB 0474

Cat. No. 2715

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Alternative Name: 3-Phenacyl UDP disodium salt

Chemical Name: 3-(2-Oxo-2-phenylethyl)-uridine-5'-diphosphate disodium salt

Biological Activity

Potent and selective P2Y₆ receptor agonist (EC₅₀ values are 70, > 1000 and > 10000 nM for P2Y₆, P2Y₂ and P2Y₄ receptors respectively).

Technical Data

M.Wt:

566.26

Formula:

C₁₇H₁₈N₂Na₂O₁₃P₂

Solubility:

Soluble in water (supplied pre-dissolved at a concentration of 10mM)

Purity:

>98 %

Storage:

Store at -20°C

CAS No:

917567-60-3

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Resources

Certificate of Analysis / Safety Data Sheet

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Safety Data Sheet: View Safety Data Sheet

References

El-Tayeb et al (2006) Synthesis and structure-activity relationships of uracil nucleotide derivatives and analogues as agonists at human P2Y₂, P2Y₄ and P2Y₆ receptors. J.Med.Chem. 49 7076. PMID: 17125260.

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