R&D Systems Inc. Tocris Bioscience Boston Biochem

O-2545 hydrochloride

Cat. No. 2680

O-2545 hydrochloride C26H36N2O2.HCl [874745-42-3]

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Chemical Name: (6aR,10aR)-6a,7,10,10a-Tetrahydro-3­-[5-(1H-imidazol-1-yl)-1,1-dimethylpentyl]-6,6,9-t­rimethyl-6H-dibenzo[b,d]pyran-1-ol hydrochloride

Biological Activity

High affinity, water-soluble CB1/CB2 receptor agonist (Ki values are 1.5 and 0.32 nM for CB1 and CB2 receptors respectively). Active in vivo following i.v. and i.c.v. administration.

Licensing Information

Sold under license from VCU-IPF

Technical Data

M.Wt:
445.04
Formula:
C26H36N2O2.HCl
Solubility:
Soluble to 100 mM in water and to 100 mM in ethanol
Purity:
>99 %
Storage:
Store at -20°C
CAS No:
874745-42-3

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Resources

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

References

Martin et al (2006) Pharmacological characterization of novel water-soluble cannabinoids. J.Pharmacol.Exp.Ther. 318 1230. PMID: 16757541.

If you know of a relevant citation for this product please let us know.

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