Cat. No. 1584
Chemical Name: N-(4-Acetylphenyl)-2-[4-(2,3,6,7-te
Biological ActivityPotent and selective adenosine A2B receptor inverse agonist (Ki values are 1.39, 157, 112 and 230 nM for human A2B, A1, A2A and A3 receptors respectively).
Licensing InformationManufactured and sold under license from Adenosine Therapeutics, LLC
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Kim et al (2000) Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A2B adenosine receptors. J.Med.Chem. 43 1165. PMID: 10737749.
Kiec-Kononowicz et al (2001) New developments in A1 and A2 adenosine receptor antagonists. Pure Appl.Chem. 73 1411.
Li et al (2007) ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor. J.Pharmacol.Exp.Ther. 320 637. PMID: 17077318.
If you know of a relevant citation for this product please let us know.
Keywords: MRS 1706, supplier, Potent, selective, A2B, inverse, agonists, Receptors, adenosines, MRS1706
Find multiple products by catalog number
New Products in this Area
Potent adenosine A2A and A2B receptor partial agonistIstradefylline
Potent and selective adenosine A2A receptor antagonistTC-G 1004
Potent and selective A2A antagonistPSB 0777 ammonium salt
Potent adenosine A2A agonist
Win a Kindle Fire HD
April 5 - 9, 2014
San Diego CA, USA
Booth Number: 2610