Nalmefene d3Cat No.
3971
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Price and Availability |
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Chemical Name: (5a)-17-(d3-Cyclopropylmethyl)-4,5-epoxy-6-methylenemor phinan-3,14-diol |
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Biological Activity
Deuterated nalmefene. Opioid receptor antagonist; displays a longer half-life in vivo than naloxone (Cat. No. 0599).Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Michel et al (1985) Binding of a new opiate antagonist, nalmefene, to rat brain membranes. Methods Find.Exp.Clin.Pharmacol. 7 175. Wang et al (1998) Nalmefene: a long-acting opioid antagonist. Clinical applications in emergency medicine. J.Emerg.Med. 16 471. Osborn et al (2010) In vivo characterization of the opioid antagonist nalmefene in mice. Life Sci. 86 624.If you know of a useful citation for this product please let us know.
Keywords: Nalmefene d3, opioid, receptors, antagonists
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