Meptazinol hydrochlorideCat No. 3636 |
Price and Availability |
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Chemical Name: 3-(3-Ethylhexahydro-1-methyl-1H-azepin-3-yl)phenol hydrochloride |
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Biological Activity
Centrally active opioid analgesic. Partial agonist at the μ1 opioid receptor. Also shown to inhibit acetylcholinesterase.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Spiegel and Pasternak (1984) Meptazinol: a novel Mu-1 selective opioid analgesic. J.Pharmacol.Exp.Ther. 228 414. Galli et al (1996) Reversible inhibition of cholinesterases by opioids: possible pharmacological consequences. J.Pharm.Pharmacol. 48 1164If you know of a useful citation for this product please let us know.
Keywords: Meptazinol hydrochloride, Partial, agonists, μ1-opioid, mu1-opioid, Receptors, MOP, Receptors, OP3, μ-opioid, mu-opioid
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