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M 1145

Cat No. 3629

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Biological Activity

Potent and selective galanin receptor 2 (GAL₂) agonist (EC₅₀ = 38 nM, K_i values are 6.55, 497 and 587 nM at GAL₂, GAL₃ and GAL₁ respectively). Has an additive effect on the signal transduction of galanin.

Technical Data

M.Wt:

2774.26

Formula:

C₁₂₈H₂₀₅N₃₇O₃₂

Sequence:

RGRGNWTLNSAGYLLGPVLPPPALALA

(Modifications: Ala-27 = C-terminal amide)

Storage:

Desiccate at -20°C

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.

Resources

Certificate of Analysis / MSDS

Certificate of Analysis: View current batch

Material Safety Data Sheet: View current batch

References

Runesson et al (2009) A novel GalR2-specific peptide agonist. Neuropeptides 43 187.

If you know of a useful citation for this product please let us know.

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Keywords: M 1145, Potent, selective, GAL2, GalR2, agonists, Receptors, Galanin

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