Tizanidine hydrochlorideCat No. 3609 |
Price and Availability |
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Chemical Name: 5-(Chloro-N-(4,5-dihydro-1H-imidazol-2-yl)-2,1,3-benzot hiadiazol-4-amine hydrochloride |
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Biological Activity
α2-adrenergic receptor agonist. Antinociceptive upon epidural administration in rats (IC50 = 48 nM). Also binds to imidazoline receptor.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis and MSDS.
Resources
Certificate of Analysis / MSDS
References
Asano et al (2000) Antinociception by epidural and systemic a2-adrenoceptor agonists and their binding affinity in rat spinal cord and brain. Anesth.Analg. 90 400. Piletz et al (2000) Autoradiographic comparison of [3H]-Clonidine binding to non-adrenergic sites and a2-adrenergic receptors in human brain. Neuropsychopharmacology 23 697.If you know of a useful citation for this product please let us know.
Keywords: Tizanidine hydrochloride, α2-Adrenergic, alpha2-Adrenergic, a2-adrenergic, α2-adrenoceptor, alpha2-adrenoceptors, a2-adrenoceptors, agonists, Receptors
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