R&D Systems Inc. Tocris Bioscience Boston Biochem

Estropipate

Cat. No. 3588

Estropipate C18H22O5S.C4H10N2 [7280-37-7]

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Chemical Name: Piperazine estrone sulfate

Biological Activity

Estrogen receptor agonist. Also inhibits organic anion transporting polypeptide 1B1 (OATP1B1) (IC50= 70 nM).

Technical Data

M.Wt:
436.56
Formula:
C18H22O5S.C4H10N2
Solubility:
Soluble to 5 mM in water and to 100 mM in DMSO
Purity:
>97 %
Storage:
Store at RT
CAS No:
7280-37-7

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

References

Williams et al (2004) Estrogen regulation of the cytochrome P450 3A subfamily in humans. J.Pharmacol.Exp.Ther. 311 728. PMID: 15282264.

Obaidat et al (2009) A cell-based high-throughput assay to identify inhibitors of organic anion transporting polypeptides 1B1 and 1B3. FASEB J. 23 748.

If you know of a relevant citation for this product please let us know.

View Related Products by Target

Keywords: Estropipate, supplier, Estrogen, receptor, agonists, OATP1B, inhibitors

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