Cat. No. 3247
Alternative Name: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Biological ActivityPotent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113. PMID: 7475964.
Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233. PMID: 12738037.
Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054. PMID: 14557380.
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Keywords: Fentanyl citrate, supplier, Potent, selective, μ-opioid, mu-opioid, agonists, MOP, Receptors, OP3
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