R&D Systems Inc. Tocris Bioscience Boston Biochem

Cannabigerol

Cat. No. 3021

Cannabigerol C21H32O2 [25654-31-3]

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Chemical Name: 2-[(2E)-3,7-Dimethyl-2,6-octadienyl­)-5-pentyl-1,3-benzenediol

Biological Activity

Partial agonist of CB2 and CB1 receptors (Ki values are 337 and 440 nM respectively). Also exhibits α2-adrenoceptor agonist activity (EC50 = 0.2 nM in mouse brain membranes).

Technical Data

M.Wt:
316.48
Formula:
C21H32O2
Solubility:
Soluble to 100 mM in ethanol and to 100 mM in DMSO
Purity:
>99 %
Storage:
Store at -20°C
CAS No:
25654-31-3

The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.

Resources

Certificate of Analysis / Safety Data Sheet

Certificate of Analysis: View current batch
Safety Data Sheet: View Safety Data Sheet

References

Pertwee The diverse CB1 and CB2 receptor pharmacology of three plant cannabinoids: Δ9-tetrahydrocannabinol, cannabidiol and Δ9-tetrahydrocannabivarin. Br.J.Pharmacol. 153 199. PMID: 17828291.

Gauson et al (2007) Cannabigerol behaves as a partial agonist at both CB1 and CB2 receptors. Symposium on the Cannabinoids 206.

Cascio et al (2010) Evidence that the plant cannabinoid cannabigerol is a highly potent α2-adrenoceptor agonist and moderately potent 5HT1A receptor antagonist. Br.J.Pharmacol. 159 129. PMID: 20002104.

If you know of a relevant citation for this product please let us know.

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