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MetaphitCat. No. 0568 |
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Chemical Name: 1-(1-(3-Isothiocyanato)phenyl)cyclohexylpiperidine |
Biological Activity
Acylator of PCP and σ-receptors.Technical Data
M.Wt:The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Certificate of Analysis / Safety Data Sheet
References
Rafferty et al (1985) A specific acylating agent for the [3H]-phencyclidine receptors in rat brain. FEBS Lett. 181 318. PMID: 2982662.
Contreras et al (1986) Metaphit, an acylating ligand for phencyclidine receptors: characterization of in vivo actions in the rat. J.Pharmacol.Exp.Ther. 238 1101. PMID: 3018219.
Debler et al (1989) Metaphit, an isothiocyanate analog of PCP, induces audiogenic seizures in mice. Eur.J.Pharmacol. 165 155. PMID: 2548879.
Reith et al (1991) Effect of metaphit on dopaminergic neurotransmission in rat striatal slices: involvement of the dopamine transporter and voltage-dependent sodium channel. J.Pharmacol.Exp.Ther. 259 1188. PMID: 1662274.
If you know of a relevant citation for this product please let us know.
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Keywords: Metaphit, supplier, Acylator, PCP, σ, sigma, receptors
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