GR 135531

Cat. No. 0896

GR 135531 C14H17N3O3 [190277-13-5]

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Alternative Name: 5-MCA-NAT

Chemical Name: 5-Methoxycarbonylamino-N-acetyltryptamine

Biological Activity

Binds with high affinity to MT3 melatonin sites in hamster brain, and low affinity (and no efficacy) at MT1 and MT2 melatonin receptors and thus can be used to discriminate between the melatonin receptor subtypes.

Technical Data

Soluble to 100 mM in ethanol
>97 %
Store at RT

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.

Certificate of Analysis / Safety Data Sheet

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Dubocovich (1995) Melatonin receptors: are there multiple subtypes? TiPS 16 50. PMID: 7762083.

Lucchelli et al (1997) Investigation into the contractile response of melatonin in the guinea-pig isolated proximal colon: the role of 5-HT4 and melatonin receptors. Br.J.Pharmacol. 121 1775. PMID: 9283717.

If you know of a relevant citation for this product please let us know.

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Keywords: GR 135531, supplier, High, affinity, melatonin, MT3, ligands, Receptors, GR135531, 5MCANAT, Melatonin Receptor Ligands

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