All Products

Cat.No.

Product Name / Activity

Potent, selective BTK inhibitor

Potent, selective mGlu_8a agonist

5-Lipoxygenase inhibitor

Selective inhibitor of mitotic kinesin Eg5

Selective PPARγ agonist

Selective, competitive nociceptin antagonist

Potent, selective P2X₁ antagonist

Highly potent blocker of K_Ca2

Inhibitor of 5-lipoxygenase-activating protein (FLAP)

Selective PPARα agonist

Selective blocker of inward-rectifier K⁺ channels

Potent, selective 5-HT_1B agonist

Potent, selective CB₁ agonist

Potent, highly selective CB₁ agonist

Potent, selective c-Raf inhibitor

Potent, selective 5-HT₄ antagonist

CCK-inactivating serine protease inhibitor

Potent, selective α_2D antagonist

Potent, subtype-selective α_1A antagonist

PPARγ antagonist

Selective for α5-containing GABA_A receptors

Benzodiazepine antagonist

Ca²⁺ release inhibitor

Cell-permeable protein kinase C inhibitor

EGFR, p60^c-src inhibitor

Cell-permeable cAMP analog

H⁺-ATPase (vacuolar) inhibitor

Protein phosphatase 1 and 2A inhibitor

cAMP antagonist

Endogenous CB receptor agonist

Potent α3β2 and β3 subunit selective nicotinic antagonist

Selective CB₂ agonist

Potent CB₁ and CB₂ agonist

Potent, selective CB₂ agonist

AMP-activated protein kinase substrate

Potent M₂/M₄ antagonist

Endogenous ghrelin receptor ligand

Highly potent, preferential D₃ antagonist

Subunit selective nAChR agonist

PDE4 inhibitor. More active enantiomer of rolipram (Cat. No. 0905)

PDE4 inhibitor. Less active enantiomer of rolipram (Cat. No. 0905)

Glycogen synthase kinase-3 substrate (synthetic)

Akt/PKB substrate (synthetic)

Potent CB₁ and TRPV1 agonist. Also anandamide transport inhibitor

Potent K_ir6 (K_ATP) channel opener

α7 neuronal nicotinic receptor antagonist

Potent, selective D₃ antagonist

Potent ORL₁ agonist

Potent, selective hA₃ antagonist

Potent, selective non-peptide AT₂ antagonist

Potent, silent TRPV1 antagonist

Allosteric potentiator of A₁ receptors

Inhibitor of tubulin

Potent, selective NPY Y₅ agonist

Potent, selective JAK3 inhibitor

Potent, selective JAK3 inhibitor

Selective Hsp90 inhibitor

Group III mGlu antagonist

Endogenous agonist at S1P_1-5

5-HT_2C/2B antagonist

Potent, selective 5-HT_2B antagonist

Potent and selective 5-HT₄ antagonist

5-HT_2C/2B antagonist/inverse agonist

Potent, selective non-peptide NK₃ antagonist

K_ir6 (K_ATP) channel opener

K_ir6 (K_ATP) channel opener. Active enantiomer of cromakalim (Cat. No. 1377)

Potent, selective 5-HT_2C/2B antagonist

GCP II inhibitor

Potent, selective c-Raf1 kinase inhibitor

Potent, selective non-peptide NPY Y₅ receptor antagonist

Potent, selective CB₂ ligand

Selective M₁ muscarinic agonist

Potent, highly selective hA₃ antagonist

Potent, highly selective VPAC₁ agonist

Potent, selective NOP partial agonist peptide

Potent, selective neuronal nicotinic agonist

Highly selective P2X₁ antagonist

Potent, selective anandamide transport inhibitor

Potent, selective non-peptide NK₃ antagonist. Brain penetrant

Potent systemically active anticonvulsant. Racemate of (R)-3,4,-DCPG (Cat. No. 1395)

AMPA antagonist/weak NMDA antagonist

Synthetic retinoid. Potent anticancer agent

Potent, selective Src inhibitor

Potent cyclin-dependent kinase inhibitor. Also inhibits GSK-3

Non-peptide, potent K_V1.3 channel blocker