All Products

Cat.No.

Product Name / Activity

Benzodiazepine inverse agonist, putative endogenous ligand

Potent and selective 5-HT_1A partial agonist

Potent 5-HT_1A ligand

EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor

PDE4 inhibitor

Inhibits K⁺ outward/pacemaker current

Selective GABA_B agonist

Potent dopamine uptake inhibitor

Selective DA uptake inhibitor. Also σ ligand

Nicotinic antagonist

α₂ agonist

High affinity σ ligand

Selective D₂-like agonist

Protein kinase C activator

Myosin light chain kinase inhibitor

PDE5 inhibitor

Protein kinase C activator

β agonist

PDE4 inhibitor

A₁ selective antagonist

Potent and specific 5-HT₃ agonist

Urokinase inhibitor

Melatonin agonist

Dopamine antagonist with some D₄ selectivity. Also 5-HT_2A/2C antagonist

Calpain and cathepsin L inhibitor

Oxidative phosphorylation uncoupler

Oxidative phosphorylation uncoupler

High affinity σ₁ ligand

Aromatic L-amino acid decarboxylase inhibitor

Skeletal muscle relaxant

5-HT re-uptake inhibitor

5-HT₁ agonist. Also has high affinity for 5-ht_5a and 5-HT₇

Selective 5-HT₂ antagonist

Prototypic vanilloid receptor agonist

Vanilloid receptor antagonist. Also activator of ENaCδ

Spermine and spermidine acetyltransferase potentiator

Muscarinic antagonist, M₁ > M₂

Standard selective κ agonist. Less active enantiomer of (±)-U-50488 (Cat. No. 0495)

Partial α agonist. Non-selective

Partial α agonist. Non-selective

Inhibits tetrahydrobiopterin synthesis and thus NOS activity

Intermediate in lipid metabolism

Urease inhibitor

Oxidative phosphorylation uncoupler

Adenosine uptake inhibitor

Muscarinic M₃ antagonist

Catechol O-methyltransferase inhibitor

Diacylglycerol kinase inhibitor

Aldose reductase inhibitor

A₁ selective antagonist

EGFR/PDGFR-kinase inhibitor

Standard selective κ agonist

Standard selective κ agonist. More active enantiomer of (±)-U-50488 (Cat. No. 0495)

EGFR-kinase inhibitor

κ agonist